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Naltrexone belongs to a class of drugs known as opiate antagonists. It works in the brain to prevent opiate effects (e.g., feelings of well-being, pain relief). It also decreases the desire to take opiates. This medication is also used to treat alcohol abuse.
In terms of dosing, 50mg of naltrexone have the ability to block the effects of opioids for about 24 hours. Clinical studies suggest that doubling the dose will block opioid effects for 48 hours, while 150mg of naltrexone can provide blockage for approximately 72 hours.
Naltrexone is a medication that blocks the effects of drugs known as opioids (a class that includes morphine, heroin or codeine). It competes with these drugs for opioid receptors in the brain. … Second, naltrexone helps patients remain abstinent.
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No, you cannot get high on naltrexone. In fact, naltrexone is prescribed to treat opiate/opioid addiction and alcoholism by blocking the pleasurable and euphoric effects of these substances. It works by binding to opioid receptors in the central nervous system that these drugs normally occupy.
Low-dose naltrexone (LDN) describes the off-label use of the medication naltrexone at low doses for diseases such as multiple sclerosis. Naltrexone is typically prescribed for opioid dependence or alcohol dependence, as it is a strong opioid antagonist. -
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